Sfoglia per Autore
Synthesis, in Vitro, and in Cell Studies of a New Series of [Indoline-3,2 '-thiazolidine]-Based p53 Modulators
2013 Bertamino, A; Soprano, M; Musella, S; Rusciano, Mr; Sala, M; Vernieri, E; Di Sarno, V; Limatola, A; Carotenuto, A; Cosconati, Sandro; Grieco, P; Novellino, E; Illario, M; Campiglia, P; Gomez Monterrey, I.
The G-triplex DNA
2013 Limongelli, V; De Tito, S; Cerofolini, L; Fragai, M; Pagano, B; Trotta, R; Cosconati, Sandro; Marinelli, L; Novellino, E; Bertini, I; Randazzo, A; Luchinat, C; Parrinello, M.
Exploring the chemical space of G-quadruplex binders: Discovery of a novel chemotype targeting the human telomeric sequence
2013 Di Leva, Fs; Zizza, P; Cingolani, C; D'Angelo, C; Pagano, B; Amato, J; Salvati, E; Sissi, C; Pinato, O; Marinelli, L; Cavalli, A; Cosconati, Sandro; Novellino, E; Randazzo, A; Biroccio, A.
Tuning RNA Interference by Enhancing siRNA/PAZ Recognition
2013 Gaglione, M; Potenza, Nicoletta; Di Fabio, G; Romanucci, V; Mosca, N; Russo, Aniello; Novellino, E; Cosconati, Sandro; Messere, Anna
Human recombinant beta-secretase immobilized enzyme reactor for fast hits' selection and characterization from a virtual screening library
2013 De Simone, A; Mancini, F; Cosconati, Sandro; Marinelli, L; La Pietra, V; Novellino, E; Andrisano, V.
Ligand based approach to L-type calcium channel by imidazo[2,1-b]thiazole- 1,4-dihydropyridines: From heart activity to brain affinity
2013 Locatelli, A; Cosconati, Sandro; Micucci, M; Leoni, A; Marinelli, L; Bedini, A; Ioan, P; Spampinato, Sm; Novellino, E; Chiarini, A; Budriesi, R.
Revisiting a Receptor-Based Pharmacophore Hypothesis for Human A(2A) Adenosine Receptor Antagonists
2013 Bacilieri, M; Ciancetta, A; Paoletta, S; Federico, S; Cosconati, Sandro; Cacciari, B; Taliani, S; Da Settimo, F; Novellino, E; Klotz, Kn; Spalluto, G; Moro, S.
tert-Butylcarbamate-Containing Histone Deacetylase Inhibitors: Apoptosis Induction, Cytodifferentiation, and Antiproliferative Activities in Cancer Cells
2013 Valente, S; Trisciuoglio, D; Tardugno, M; Benedetti, R; Labella, D; Secci, D; Mercurio, C; Boggio, R; Tomassi, S; DI MARO, Salvatore; Novellino, E; Altucci, Lucia; Del Bufalo, D; Mai, A; Cosconati, Sandro
Phenylpyrazolo[1,5-a]quinazolin-5(4 H)-one: A suitable scaffold for the development of noncamptothecin topoisomerase i (Top1) inhibitors
2013 Taliani, S; Pugliesi, I; Barresi, E; Salerno, S; Marchand, C; Agama, K; Simorini, F; La Motta, C; Marini, Am; Di Leva, Fs; Marinelli, L; Cosconati, Sandro; Novellino, E; Pommier, Y; Di Santo, R; Da Settimo, F.
Inhibition of Ocular Aldose Reductase by a New Benzofuroxane Derivative Ameliorates Rat Endotoxic Uveitis
2014 DI FILIPPO, Clara; Zippo, Mv; Maisto, R; Trotta, Mc; Siniscalco, D; Ferraro, B; Ferraraccio, Franca; La Motta, C; Sartini, S; Cosconati, Sandro; Novellino, E; Gesualdo, C; Simonelli, Francesca; Rossi, Settimio; D'Amico, Michele
Identification of highly conserved residues involved in inhibition of HIV-1 RNase H function by diketo acid derivatives
2014 Corona, A; Di Leva, Fs; Thierry, S; Pescatori, L; Cuzzucoli Crucitti, G; Subra, F; Delelis, O; Esposito, F; Rigogliuso, G; Costi, R; Cosconati, Sandro; Novellino, E; Di Santo, R; Tramontano, E.
Properly Substituted Analogues of BIX-01294 Lose Inhibition of G9a Histone Methyltransferase and Gain Selective Anti-DNA Methyltransferase 3A Activity
2014 Rotili, D; Tarantino, D; Marrocco, B; Gros, C; Masson, V; Poughon, V; Ausseil, F; Chang, Y; Labella, D; Cosconati, Sandro; DI MARO, Salvatore; Novellino, E; Schnekenburger, M; Grandjenette, C; Bouvy, C; Diederich, M; Cheng, X; Arimondo, Pb; Mai, A.
Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase
2014 Costi, R; Metifiot, M; Chung, S; Crucitti, Gv; Maddali, K; Pescatori, L; Messore, A; Madia, Vn; Pupo, G; Scipione, L; Tortorella, S; Di Leva, Fs; Cosconati, Sandro; Marinelli, L; Novellino, E; Le Grice, Sfj; Corona, A; Pommier, Y; Marchand, C; Di Santo, R.
Shading the TRF2 Recruiting Function: A New Horizon in Drug Development
2014 DI MARO, Salvatore; Zizza, P; Salvati, E; De Luca, V; Capasso, C; Fotticchia, I; Pagano, B; Marinelli, L; Gilson, E; Novellino, E; Cosconati, Sandro; Biroccio, A.
Structure-Activity Relationship Refinement and Further Assessment of 4-Phenylquinazoline-2-carboxamide Translocator Protein Ligands as Antiproliferative Agents in Human Glioblastoma Tumors
2014 Castellano, S; Taliani, S; Viviano, M; Milite, C; Da Pozzo, E; Costa, B; Barresi, E; Bruno, A; Cosconati, Sandro; Marinelli, L; Greco, G; Novellino, E; Sbardella, G; Da Settimo, F; Martini, C.
Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells
2014 Valente, S; Liu, Y; Schnekenburger, M; Zwergel, C; Cosconati, Sandro; Gros, C; Tardugno, M; Labella, D; Florean, C; Minden, S; Hashimoto, H; Chan, Y; Zhang, X; Kirsch, G; Novellino, E; Arimondo, Pb; Miele, E; Ferretti, E; Gulino, A; Diederich, M; Cheng, X; Mai, A.
Synthesis and gene silencing properties of siRNAs containing terminal amide linkages
2014 Gaglione, M; Mercurio, Me; Potenza, Nicoletta; Mosca, N; Russo, Aniello; Novellino, E; Cosconati, Sandro; Messere, Anna
The first sphingosine 1-phosphate lyase inhibitors against multiple sclerosis: A successful drug discovery tale
2014 Cosconati, Sandro; Novellino, E.
Discovery of N-aryl-naphthylamines as in vitro inhibitors of the interaction between HIV integrase and the cofactor LEDGF/p75
2015 Cuzzucoli Crucitti, G; Pescatori, L; Messore, A; Madia, Vn; Pupo, G; Saccoliti, F; Scipione, L; Tortorella, S; Di Leva, Fs; Cosconati, Sandro; Novellino, E; Debyser, Z; Christ, F; Costi, R; Di Santo, R.
Endogenous vs Exogenous Allosteric Modulators in GPCRs: A dispute for shuttling CB1 among different membrane microenvironments
2015 Stornaiuolo, Mariano; Bruno, Agostino; Botta, Lorenzo; Regina, Giuseppe La; Cosconati, Sandro; Silvestri, Romano; Marinelli, Luciana; Novellino, Ettore
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis, in Vitro, and in Cell Studies of a New Series of [Indoline-3,2 '-thiazolidine]-Based p53 Modulators | 1-gen-2013 | Bertamino, A; Soprano, M; Musella, S; Rusciano, Mr; Sala, M; Vernieri, E; Di Sarno, V; Limatola, A; Carotenuto, A; Cosconati, Sandro; Grieco, P; Novellino, E; Illario, M; Campiglia, P; Gomez Monterrey, I. | |
The G-triplex DNA | 1-gen-2013 | Limongelli, V; De Tito, S; Cerofolini, L; Fragai, M; Pagano, B; Trotta, R; Cosconati, Sandro; Marinelli, L; Novellino, E; Bertini, I; Randazzo, A; Luchinat, C; Parrinello, M. | |
Exploring the chemical space of G-quadruplex binders: Discovery of a novel chemotype targeting the human telomeric sequence | 1-gen-2013 | Di Leva, Fs; Zizza, P; Cingolani, C; D'Angelo, C; Pagano, B; Amato, J; Salvati, E; Sissi, C; Pinato, O; Marinelli, L; Cavalli, A; Cosconati, Sandro; Novellino, E; Randazzo, A; Biroccio, A. | |
Tuning RNA Interference by Enhancing siRNA/PAZ Recognition | 1-gen-2013 | Gaglione, M; Potenza, Nicoletta; Di Fabio, G; Romanucci, V; Mosca, N; Russo, Aniello; Novellino, E; Cosconati, Sandro; Messere, Anna | |
Human recombinant beta-secretase immobilized enzyme reactor for fast hits' selection and characterization from a virtual screening library | 1-gen-2013 | De Simone, A; Mancini, F; Cosconati, Sandro; Marinelli, L; La Pietra, V; Novellino, E; Andrisano, V. | |
Ligand based approach to L-type calcium channel by imidazo[2,1-b]thiazole- 1,4-dihydropyridines: From heart activity to brain affinity | 1-gen-2013 | Locatelli, A; Cosconati, Sandro; Micucci, M; Leoni, A; Marinelli, L; Bedini, A; Ioan, P; Spampinato, Sm; Novellino, E; Chiarini, A; Budriesi, R. | |
Revisiting a Receptor-Based Pharmacophore Hypothesis for Human A(2A) Adenosine Receptor Antagonists | 1-gen-2013 | Bacilieri, M; Ciancetta, A; Paoletta, S; Federico, S; Cosconati, Sandro; Cacciari, B; Taliani, S; Da Settimo, F; Novellino, E; Klotz, Kn; Spalluto, G; Moro, S. | |
tert-Butylcarbamate-Containing Histone Deacetylase Inhibitors: Apoptosis Induction, Cytodifferentiation, and Antiproliferative Activities in Cancer Cells | 1-gen-2013 | Valente, S; Trisciuoglio, D; Tardugno, M; Benedetti, R; Labella, D; Secci, D; Mercurio, C; Boggio, R; Tomassi, S; DI MARO, Salvatore; Novellino, E; Altucci, Lucia; Del Bufalo, D; Mai, A; Cosconati, Sandro | |
Phenylpyrazolo[1,5-a]quinazolin-5(4 H)-one: A suitable scaffold for the development of noncamptothecin topoisomerase i (Top1) inhibitors | 1-gen-2013 | Taliani, S; Pugliesi, I; Barresi, E; Salerno, S; Marchand, C; Agama, K; Simorini, F; La Motta, C; Marini, Am; Di Leva, Fs; Marinelli, L; Cosconati, Sandro; Novellino, E; Pommier, Y; Di Santo, R; Da Settimo, F. | |
Inhibition of Ocular Aldose Reductase by a New Benzofuroxane Derivative Ameliorates Rat Endotoxic Uveitis | 1-gen-2014 | DI FILIPPO, Clara; Zippo, Mv; Maisto, R; Trotta, Mc; Siniscalco, D; Ferraro, B; Ferraraccio, Franca; La Motta, C; Sartini, S; Cosconati, Sandro; Novellino, E; Gesualdo, C; Simonelli, Francesca; Rossi, Settimio; D'Amico, Michele | |
Identification of highly conserved residues involved in inhibition of HIV-1 RNase H function by diketo acid derivatives | 1-gen-2014 | Corona, A; Di Leva, Fs; Thierry, S; Pescatori, L; Cuzzucoli Crucitti, G; Subra, F; Delelis, O; Esposito, F; Rigogliuso, G; Costi, R; Cosconati, Sandro; Novellino, E; Di Santo, R; Tramontano, E. | |
Properly Substituted Analogues of BIX-01294 Lose Inhibition of G9a Histone Methyltransferase and Gain Selective Anti-DNA Methyltransferase 3A Activity | 1-gen-2014 | Rotili, D; Tarantino, D; Marrocco, B; Gros, C; Masson, V; Poughon, V; Ausseil, F; Chang, Y; Labella, D; Cosconati, Sandro; DI MARO, Salvatore; Novellino, E; Schnekenburger, M; Grandjenette, C; Bouvy, C; Diederich, M; Cheng, X; Arimondo, Pb; Mai, A. | |
Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase | 1-gen-2014 | Costi, R; Metifiot, M; Chung, S; Crucitti, Gv; Maddali, K; Pescatori, L; Messore, A; Madia, Vn; Pupo, G; Scipione, L; Tortorella, S; Di Leva, Fs; Cosconati, Sandro; Marinelli, L; Novellino, E; Le Grice, Sfj; Corona, A; Pommier, Y; Marchand, C; Di Santo, R. | |
Shading the TRF2 Recruiting Function: A New Horizon in Drug Development | 1-gen-2014 | DI MARO, Salvatore; Zizza, P; Salvati, E; De Luca, V; Capasso, C; Fotticchia, I; Pagano, B; Marinelli, L; Gilson, E; Novellino, E; Cosconati, Sandro; Biroccio, A. | |
Structure-Activity Relationship Refinement and Further Assessment of 4-Phenylquinazoline-2-carboxamide Translocator Protein Ligands as Antiproliferative Agents in Human Glioblastoma Tumors | 1-gen-2014 | Castellano, S; Taliani, S; Viviano, M; Milite, C; Da Pozzo, E; Costa, B; Barresi, E; Bruno, A; Cosconati, Sandro; Marinelli, L; Greco, G; Novellino, E; Sbardella, G; Da Settimo, F; Martini, C. | |
Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells | 1-gen-2014 | Valente, S; Liu, Y; Schnekenburger, M; Zwergel, C; Cosconati, Sandro; Gros, C; Tardugno, M; Labella, D; Florean, C; Minden, S; Hashimoto, H; Chan, Y; Zhang, X; Kirsch, G; Novellino, E; Arimondo, Pb; Miele, E; Ferretti, E; Gulino, A; Diederich, M; Cheng, X; Mai, A. | |
Synthesis and gene silencing properties of siRNAs containing terminal amide linkages | 1-gen-2014 | Gaglione, M; Mercurio, Me; Potenza, Nicoletta; Mosca, N; Russo, Aniello; Novellino, E; Cosconati, Sandro; Messere, Anna | |
The first sphingosine 1-phosphate lyase inhibitors against multiple sclerosis: A successful drug discovery tale | 1-gen-2014 | Cosconati, Sandro; Novellino, E. | |
Discovery of N-aryl-naphthylamines as in vitro inhibitors of the interaction between HIV integrase and the cofactor LEDGF/p75 | 1-gen-2015 | Cuzzucoli Crucitti, G; Pescatori, L; Messore, A; Madia, Vn; Pupo, G; Saccoliti, F; Scipione, L; Tortorella, S; Di Leva, Fs; Cosconati, Sandro; Novellino, E; Debyser, Z; Christ, F; Costi, R; Di Santo, R. | |
Endogenous vs Exogenous Allosteric Modulators in GPCRs: A dispute for shuttling CB1 among different membrane microenvironments | 1-gen-2015 | Stornaiuolo, Mariano; Bruno, Agostino; Botta, Lorenzo; Regina, Giuseppe La; Cosconati, Sandro; Silvestri, Romano; Marinelli, Luciana; Novellino, Ettore |
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