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Titolo Data di pubblicazione Autore(i) File
New 2-Heterocyclyl-imidazo[2,1-i]purin-5-one Derivatives as Potent and Selective Human A(3) Adenosine Receptor Antagonists 1-gen-2011 Baraldi, Pg; Preti, D; Zaid, An; Saponaro, G; Tabrizi, Ma; Baraldi, S; Romagnoli, R; Moorman, Ar; Varani, K; Cosconati, Sandro; DI MARO, Salvatore; Marinelli, L; Novellino, E; Borea, Pa
Increasing αvβ3 selectivity of the anti-angiogenic drug cilengitide by N-methylation 1-gen-2011 Mas Moruno, C; Beck, Jg; Doedens, L; Frank, Ao; Marinelli, L; Cosconati, Sandro; Novellino, E; Kessler, H.
Identification of 5-arylidene-4-thiazolidinone derivatives endowed with dual activity as aldose reductase inhibitors and antioxidant agents for the treatment of diabetic complications 1-gen-2011 Ottana, R; Maccari, R; Giglio, M; Del Corso, A; Cappiello, M; Mura, U; Cosconati, Sandro; Marinelli, L; Novellino, E; Sartini, S; La Motta, C; Da Settimo, F.
3-(Fur-2-yl)-10-(2-phenylethyl)-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)- one, a novel adenosine receptor antagonist with A2A-mediated neuroprotective effects 1-gen-2011 Scatena, A; Fornai, F; Trincavelli, Ml; Taliani, S; Daniele, S; Pugliesi, I; Cosconati, Sandro; Martini, C; Da Settimo, F.
A more detailed picture of the interactions between virtual screening-derived hits and the DNA G-quadruplex: NMR, molecular modelling and ITC studies 1-gen-2011 Trotta, R; De Tito, S; Lauri, I; La Pietra, V; Marinelli, L; Cosconati, Sandro; Martino, L; Conte, Mr; Mayol, L; Novellino, E; Randazzo, A.
Design, synthesis, and functionalization of dimeric peptides targeting chemokine receptor CXCR4 1-gen-2011 Demmer, O; Dijkgraaf, I; Schumacher, U; Marinelli, L; Cosconati, Sandro; Gourni, E; Wester, Hj; Kessler, H.
Sampling protein motion and solvent effect during ligand binding 1-gen-2012 Limongelli, V; Marinelli, L; Cosconati, Sandro; La Motta, C; Sartini, S; Mugnaini, L; Da Settimo, F; Novellino, E; Parrinello, M.
Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein 1-gen-2012 Castellano, S; Taliani, S; Milite, C; Pugliesi, I; Da Pozzo, E; Rizzetto, E; Bendinelli, S; Costa, B; Cosconati, Sandro; Greco, G; Novellino, E; Sbardella, G; Stefancich, G; Martini, C; Da, Settimo
Water-soluble pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines as human A 3 adenosine receptor antagonists 1-gen-2012 Baraldi, Pg; Saponaro, G; Romagnoli, R; Aghazadeh Tabrizi, M; Baraldi, S; Moorman, Ar; Cosconati, Sandro; DI MARO, Salvatore; Marinelli, L; Gessi, S; Merighi, S; Varani, K; Borea, Pa; Preti, D.
A conformationally frozen peptoid boosts CXCR4 affinity and anti-HIV activity 1-gen-2012 Demmer, O; Frank, Ao; Hagn, F; Schottelius, M; Marinelli, L; Cosconati, Sandro; Brack Werner, R; Kremb, S; Wester, Hj; Kessler, H.
New nitrogen containing substituents at the indole-2-carboxamide yield high potent and broad spectrum indolylarylsulfone HIV-1 non-nucleoside reverse transcriptase inhibitors 1-gen-2012 La Regina, G; Coluccia, A; Brancale, A; Piscitelli, F; Famiglini, V; Cosconati, Sandro; Maga, G; Samuele, A; Gonzales, E; Clotet, B; Schols, D; Este, J; Novellino, E; Silvestri, S.
Benzofuroxane derivatives as multi-effective agents for the treatment of cardiovascular diabetic complications. Synthesis, functional evaluation, and molecular modeling studies 1-gen-2012 Sartini, S; Cosconati, Sandro; Marinelli, M; Barresi, E; DI MARO, Salvatore; Simorini, F; Taliani, S; Salerno, S; Marini, Am; Da Settimo, F; Novellino, E; La Motta, C.
Identification of novel molecular scaffolds for the design of MMP-13 inhibitors: A first round of lead optimization 1-gen-2012 La Pietra, V; Marinelli, L; Cosconati, Sandro; Di Leva, Fs; Nuti, E; Santamaria, S; Pugliesi, I; Morelli, M; Casalini, F; Rossello, A; La Motta, C; Taliani, S; Visse, R; Nagase, H; da Settimo, F; Novellino, E.
Shooting for selective druglike G-quadruplex binders: Evidence for telomeric DNA damage and tumor cell death 1-gen-2012 Cosconati, Sandro; Rizzo, A; Trotta, R; Pagano, B; Iachettini, S; De Tito, S; Lauri, I; Fotticchia, I; Giustiniano, M; Marinelli, L; Giancola, C; Novellino, E; Biroccio, A; Randazzo, A.
State-of-the-Art Methodologies for the Discovery and Characterization of DNA G-Quadruplex Binders 1-gen-2012 Pagano, B; Cosconati, Sandro; Gabelica, V; Petraccone, L; De Tito, S; Marinelli, L; La Pietra, V; di Leva F., S; Lauri, I; Trotta, R; Novellino, E; Giancola, C; Randazzo, A.
3-Aryl-[1,2,4]triazino[4,3-a ]benzimidazol-4(10 H)-one: A novel template for the design of highly selective A2B adenosine receptor antagonists 1-gen-2012 Taliani, S; Pugliesi, I; Barresi, E; Simorini, F; Salerno, S; La Motta, C; Marini, Am; Cosimelli, B; Cosconati, Sandro; DI MARO, Salvatore; Marinelli, L; Daniele, S; Trincavelli, Ml; Greco, G; Novellino, E; Martini, C; Da Settimo, F.
Progresses in the pursuit of aldose reductase inhibitors: The structure-based lead optimization step 1-gen-2012 Ramunno, A; Cosconati, Sandro; Sartini, S; Maglio, V; Angiuoli, S; La Pietra, V; DI MARO, Salvatore; Giustiniano, M; La Motta, C; Da Settimo, F; Marinelli, L; Novellino, E.
Synthesis and Biological Evaluation of CTP Synthetase Inhibitors as Potential Agents for the Treatment of African Trypanosomiasis 1-gen-2012 Tamborini, L; Pinto, A; Smith, Tk; Major, Ll; Iannuzzi, Mc; Cosconati, Sandro; Marinelli, L; Novellino, E; Lo Presti, L; Wong, Pe; Barrett, Mp; De Micheli, C; Conti, P.
From the Pharmacophore to the Homology Model of the Benzodiazepine Receptor: The Indolyglyoxylamides Affair 1-gen-2012 Cosimelli, B; Cosconati, Sandro; Marinelli, L; Novellino, E; Greco, G.
Protein Flexibility in Virtual Screening: The BACE-1 Case Study 1-gen-2012 Cosconati, Sandro; Marinelli, L; Di Leva, Fs; La Pietra, V; De Simone, A; Mancini, F; Andrisano, V; Novellino, E; Goodsell, D; Olson, A. J.
Mostrati risultati da 21 a 40 di 120
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