COSCONATI, Sandro
COSCONATI, Sandro
Dipartimento di Scienze e Tecnologie Ambientali Biologiche e Farmaceutiche (DISTABiF)
3-(Fur-2-yl)-10-(2-phenylethyl)-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)- one, a novel adenosine receptor antagonist with A2A-mediated neuroprotective effects
2011 Scatena, A; Fornai, F; Trincavelli, Ml; Taliani, S; Daniele, S; Pugliesi, I; Cosconati, Sandro; Martini, C; Da Settimo, F.
3-Aryl-[1,2,4]triazino[4,3-a ]benzimidazol-4(10 H)-one: A novel template for the design of highly selective A2B adenosine receptor antagonists
2012 Taliani, S; Pugliesi, I; Barresi, E; Simorini, F; Salerno, S; La Motta, C; Marini, Am; Cosimelli, B; Cosconati, Sandro; DI MARO, Salvatore; Marinelli, L; Daniele, S; Trincavelli, Ml; Greco, G; Novellino, E; Martini, C; Da Settimo, F.
4-Imidazo[2,1-b]thiazole-1,4-DHPs and neuroprotection: preliminary study in hits searching
2019 Leoni, Alberto; Frosini, Maria; Locatelli, Alessandra; Micucci, Matteo; Carotenuto, Claudio; Durante, Miriam; Cosconati, Sandro; Budriesi, Roberta
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors
2018 Salerno, Silvia; Barresi, Elisabetta; Amendola, Giorgio; Berrino, Emanuela; Milite, Ciro; Marini, Anna Maria; Da Settimo, Federico; Novellino, Ettore; Supuran, Claudiu T; Cosconati, Sandro; Taliani, Sabrina
A balance between elongation and trimming regulates telomere stability in stem cells
2017 Rivera, Teresa; Haggblom, Candy; Cosconati, Sandro; Karlseder, Jan
A conformationally frozen peptoid boosts CXCR4 affinity and anti-HIV activity
2012 Demmer, O; Frank, Ao; Hagn, F; Schottelius, M; Marinelli, L; Cosconati, Sandro; Brack Werner, R; Kremb, S; Wester, Hj; Kessler, H.
A cyanine-based NIR fluorescent Vemurafenib analog to probe BRAFV600E in cancer cells
2023 Barresi, Elisabetta; Baldanzi, Caterina; Roncetti, Marta; Roggia, Michele; Baglini, Emma; Lepori, Irene; Vitiello, Marianna; Salerno, Silvia; Tedeschi, Lorena; Da Settimo, Federico; Cosconati, Sandro; Poliseno, Laura; Taliani, Sabrina
A more detailed picture of the interactions between virtual screening-derived hits and the DNA G-quadruplex: NMR, molecular modelling and ITC studies
2011 Trotta, R; De Tito, S; Lauri, I; La Pietra, V; Marinelli, L; Cosconati, Sandro; Martino, L; Conte, Mr; Mayol, L; Novellino, E; Randazzo, A.
A novel smaller β-defensin-derived peptide is active against multidrug-resistant bacterial strains
2021 Colicchio, R.; Nigro, E.; Colavita, I.; Pagliuca, C.; Di Maro, S.; Tomassi, S.; Scaglione, E.; Carbone, F.; Carriero, M. V.; Matarese, G.; Daniele, A.; Cosconati, S.; Pessi, A.; Salvatore, F.; Salvatore, P.
A unique capsular polysaccharide structure from the psychrophilic marine bacterium Colwellia psychrerythraea 34H that mimics antifreeze (glyco)proteins
2015 Carillo, S; Casillo, A; Pieretti, G; Parrilli, E; Sannino, F; Bayer-Giraldi, M; Cosconati, S; Novellino, E; Ewert, M; Deming, Jw; Lanzetta, R; Marino, G; Parrilli, M; Randazzo, A; Tutino, Ml; Corsaro, Mm.
Antiproliferative and proapoptotic activity of CLM3, a novel multiple tyrosine kinase inhibitor, alone and in combination with SN-38 on endothelial and cancer cells
2011 Bocci, G; Fioravanti, A; La Motta, C; Orlandi, P; Canu, B; Di Desidero, T; Mugnaini, L; Sartini, S; Cosconati, Sandro; Frati, R; Antonelli, A; Berti, P; Miccoli, P; Da Settimo, F; Danesi, R.
Antitumor efficacy of Kisspeptin in human malignant mesothelioma cells
2018 Ciaramella, V; DELLA CORTE, Carminia Maria; Di Mauro, C; Tomassi, S; Di Maro, S; Troiani, T; Martinelli, E; Bianco, R; Cosconati, S; Pierantoni, R; Meccariello, R; Chianese, R; Ciardiello, F; Morgillo, F.
Architecture of the human urotensin II receptor: Comparison of the binding domains of peptide and non-peptide urotensin II agonists
2005 Lavecchia, A; Cosconati, Sandro; Novellino, E.
Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase
2014 Costi, R; Metifiot, M; Chung, S; Crucitti, Gv; Maddali, K; Pescatori, L; Messore, A; Madia, Vn; Pupo, G; Scipione, L; Tortorella, S; Di Leva, Fs; Cosconati, Sandro; Marinelli, L; Novellino, E; Le Grice, Sfj; Corona, A; Pommier, Y; Marchand, C; Di Santo, R.
Benzofuroxane derivatives as multi-effective agents for the treatment of cardiovascular diabetic complications. Synthesis, functional evaluation, and molecular modeling studies
2012 Sartini, S; Cosconati, Sandro; Marinelli, M; Barresi, E; DI MARO, Salvatore; Simorini, F; Taliani, S; Salerno, S; Marini, Am; Da Settimo, F; Novellino, E; La Motta, C.
Best Matching Protein Conformations and Docking Programs for a Virtual Screening Campaign Against SMO Receptor
2016 Amendola, Giorgio; Dimaio, Danilo; Lapietra, Valeria; Cosconati, Sandro
Boosting Fmoc Solid-Phase Peptide Synthesis by Ultrasonication
2019 Merlino, F.; Tomassi, S.; Yousif, A. M.; Messere, A.; Marinelli, L.; Grieco, P.; Novellino, E.; Cosconati, S.; Di Maro, S.
Carbonic anhydrase activation profile of indole-based derivatives
2021 Barresi, E.; Ravichandran, R.; Germelli, L.; Angeli, A.; Baglini, E.; Salerno, S.; Marini, A. M.; Costa, B.; Da Pozzo, E.; Martini, C.; Da Settimo, F.; Supuran, C.; Cosconati, S.; Taliani, S.
Cationic nucleopeptides as novel non-covalent carriers for the delivery of peptide nucleic acid (PNA) and RNA oligomers
2018 Tomassi, Stefano; Ieranò, Caterina; Mercurio, Maria Emilia; Nigro, Ersilia; Daniele, Aurora; Russo, Rosita; Chambery, Angela; Baglivo, Ilaria; Pedone, Paolo Vincenzo; Rea, Giuseppina; Napolitano, Maria; Scala, Stefania; Cosconati, Sandro; Marinelli, Luciana; Novellino, Ettore; Messere, Anna; Di Maro, Salvatore
Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic Activity
2015 Eadsforth, Tc; Pinto, A; Luciani, R; Tamborini, L; Cullia, G; De Micheli, C; Marinelli, L; Cosconati, Sandro; Novellino, E; Lo Presti, L; Cordeiro da Silva, A; Conti, P; Hunter, Wn; Costi, M. P.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
3-(Fur-2-yl)-10-(2-phenylethyl)-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)- one, a novel adenosine receptor antagonist with A2A-mediated neuroprotective effects | 1-gen-2011 | Scatena, A; Fornai, F; Trincavelli, Ml; Taliani, S; Daniele, S; Pugliesi, I; Cosconati, Sandro; Martini, C; Da Settimo, F. | |
3-Aryl-[1,2,4]triazino[4,3-a ]benzimidazol-4(10 H)-one: A novel template for the design of highly selective A2B adenosine receptor antagonists | 1-gen-2012 | Taliani, S; Pugliesi, I; Barresi, E; Simorini, F; Salerno, S; La Motta, C; Marini, Am; Cosimelli, B; Cosconati, Sandro; DI MARO, Salvatore; Marinelli, L; Daniele, S; Trincavelli, Ml; Greco, G; Novellino, E; Martini, C; Da Settimo, F. | |
4-Imidazo[2,1-b]thiazole-1,4-DHPs and neuroprotection: preliminary study in hits searching | 1-gen-2019 | Leoni, Alberto; Frosini, Maria; Locatelli, Alessandra; Micucci, Matteo; Carotenuto, Claudio; Durante, Miriam; Cosconati, Sandro; Budriesi, Roberta | |
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors | 1-gen-2018 | Salerno, Silvia; Barresi, Elisabetta; Amendola, Giorgio; Berrino, Emanuela; Milite, Ciro; Marini, Anna Maria; Da Settimo, Federico; Novellino, Ettore; Supuran, Claudiu T; Cosconati, Sandro; Taliani, Sabrina | |
A balance between elongation and trimming regulates telomere stability in stem cells | 1-gen-2017 | Rivera, Teresa; Haggblom, Candy; Cosconati, Sandro; Karlseder, Jan | |
A conformationally frozen peptoid boosts CXCR4 affinity and anti-HIV activity | 1-gen-2012 | Demmer, O; Frank, Ao; Hagn, F; Schottelius, M; Marinelli, L; Cosconati, Sandro; Brack Werner, R; Kremb, S; Wester, Hj; Kessler, H. | |
A cyanine-based NIR fluorescent Vemurafenib analog to probe BRAFV600E in cancer cells | 1-gen-2023 | Barresi, Elisabetta; Baldanzi, Caterina; Roncetti, Marta; Roggia, Michele; Baglini, Emma; Lepori, Irene; Vitiello, Marianna; Salerno, Silvia; Tedeschi, Lorena; Da Settimo, Federico; Cosconati, Sandro; Poliseno, Laura; Taliani, Sabrina | |
A more detailed picture of the interactions between virtual screening-derived hits and the DNA G-quadruplex: NMR, molecular modelling and ITC studies | 1-gen-2011 | Trotta, R; De Tito, S; Lauri, I; La Pietra, V; Marinelli, L; Cosconati, Sandro; Martino, L; Conte, Mr; Mayol, L; Novellino, E; Randazzo, A. | |
A novel smaller β-defensin-derived peptide is active against multidrug-resistant bacterial strains | 1-gen-2021 | Colicchio, R.; Nigro, E.; Colavita, I.; Pagliuca, C.; Di Maro, S.; Tomassi, S.; Scaglione, E.; Carbone, F.; Carriero, M. V.; Matarese, G.; Daniele, A.; Cosconati, S.; Pessi, A.; Salvatore, F.; Salvatore, P. | |
A unique capsular polysaccharide structure from the psychrophilic marine bacterium Colwellia psychrerythraea 34H that mimics antifreeze (glyco)proteins | 1-gen-2015 | Carillo, S; Casillo, A; Pieretti, G; Parrilli, E; Sannino, F; Bayer-Giraldi, M; Cosconati, S; Novellino, E; Ewert, M; Deming, Jw; Lanzetta, R; Marino, G; Parrilli, M; Randazzo, A; Tutino, Ml; Corsaro, Mm. | |
Antiproliferative and proapoptotic activity of CLM3, a novel multiple tyrosine kinase inhibitor, alone and in combination with SN-38 on endothelial and cancer cells | 1-gen-2011 | Bocci, G; Fioravanti, A; La Motta, C; Orlandi, P; Canu, B; Di Desidero, T; Mugnaini, L; Sartini, S; Cosconati, Sandro; Frati, R; Antonelli, A; Berti, P; Miccoli, P; Da Settimo, F; Danesi, R. | |
Antitumor efficacy of Kisspeptin in human malignant mesothelioma cells | 1-gen-2018 | Ciaramella, V; DELLA CORTE, Carminia Maria; Di Mauro, C; Tomassi, S; Di Maro, S; Troiani, T; Martinelli, E; Bianco, R; Cosconati, S; Pierantoni, R; Meccariello, R; Chianese, R; Ciardiello, F; Morgillo, F. | |
Architecture of the human urotensin II receptor: Comparison of the binding domains of peptide and non-peptide urotensin II agonists | 1-gen-2005 | Lavecchia, A; Cosconati, Sandro; Novellino, E. | |
Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase | 1-gen-2014 | Costi, R; Metifiot, M; Chung, S; Crucitti, Gv; Maddali, K; Pescatori, L; Messore, A; Madia, Vn; Pupo, G; Scipione, L; Tortorella, S; Di Leva, Fs; Cosconati, Sandro; Marinelli, L; Novellino, E; Le Grice, Sfj; Corona, A; Pommier, Y; Marchand, C; Di Santo, R. | |
Benzofuroxane derivatives as multi-effective agents for the treatment of cardiovascular diabetic complications. Synthesis, functional evaluation, and molecular modeling studies | 1-gen-2012 | Sartini, S; Cosconati, Sandro; Marinelli, M; Barresi, E; DI MARO, Salvatore; Simorini, F; Taliani, S; Salerno, S; Marini, Am; Da Settimo, F; Novellino, E; La Motta, C. | |
Best Matching Protein Conformations and Docking Programs for a Virtual Screening Campaign Against SMO Receptor | 1-gen-2016 | Amendola, Giorgio; Dimaio, Danilo; Lapietra, Valeria; Cosconati, Sandro | |
Boosting Fmoc Solid-Phase Peptide Synthesis by Ultrasonication | 1-gen-2019 | Merlino, F.; Tomassi, S.; Yousif, A. M.; Messere, A.; Marinelli, L.; Grieco, P.; Novellino, E.; Cosconati, S.; Di Maro, S. | |
Carbonic anhydrase activation profile of indole-based derivatives | 1-gen-2021 | Barresi, E.; Ravichandran, R.; Germelli, L.; Angeli, A.; Baglini, E.; Salerno, S.; Marini, A. M.; Costa, B.; Da Pozzo, E.; Martini, C.; Da Settimo, F.; Supuran, C.; Cosconati, S.; Taliani, S. | |
Cationic nucleopeptides as novel non-covalent carriers for the delivery of peptide nucleic acid (PNA) and RNA oligomers | 1-gen-2018 | Tomassi, Stefano; Ieranò, Caterina; Mercurio, Maria Emilia; Nigro, Ersilia; Daniele, Aurora; Russo, Rosita; Chambery, Angela; Baglivo, Ilaria; Pedone, Paolo Vincenzo; Rea, Giuseppina; Napolitano, Maria; Scala, Stefania; Cosconati, Sandro; Marinelli, Luciana; Novellino, Ettore; Messere, Anna; Di Maro, Salvatore | |
Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic Activity | 1-gen-2015 | Eadsforth, Tc; Pinto, A; Luciani, R; Tamborini, L; Cullia, G; De Micheli, C; Marinelli, L; Cosconati, Sandro; Novellino, E; Lo Presti, L; Cordeiro da Silva, A; Conti, P; Hunter, Wn; Costi, M. P. |