COSCONATI, Sandro

COSCONATI, Sandro  

Dipartimento di Scienze e Tecnologie Ambientali Biologiche e Farmaceutiche (DISTABiF)  

Risultati 1 - 20 di 119 (tempo di esecuzione: 0.02 secondi).
Titolo Data di pubblicazione Autore(i) File
3-(Fur-2-yl)-10-(2-phenylethyl)-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)- one, a novel adenosine receptor antagonist with A2A-mediated neuroprotective effects 1-gen-2011 Scatena, A; Fornai, F; Trincavelli, Ml; Taliani, S; Daniele, S; Pugliesi, I; Cosconati, Sandro; Martini, C; Da Settimo, F.
3-Aryl-[1,2,4]triazino[4,3-a ]benzimidazol-4(10 H)-one: A novel template for the design of highly selective A2B adenosine receptor antagonists 1-gen-2012 Taliani, S; Pugliesi, I; Barresi, E; Simorini, F; Salerno, S; La Motta, C; Marini, Am; Cosimelli, B; Cosconati, Sandro; DI MARO, Salvatore; Marinelli, L; Daniele, S; Trincavelli, Ml; Greco, G; Novellino, E; Martini, C; Da Settimo, F.
4-Imidazo[2,1-b]thiazole-1,4-DHPs and neuroprotection: preliminary study in hits searching 1-gen-2019 Leoni, Alberto; Frosini, Maria; Locatelli, Alessandra; Micucci, Matteo; Carotenuto, Claudio; Durante, Miriam; Cosconati, Sandro; Budriesi, Roberta
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors 1-gen-2018 Salerno, Silvia; Barresi, Elisabetta; Amendola, Giorgio; Berrino, Emanuela; Milite, Ciro; Marini, Anna Maria; Da Settimo, Federico; Novellino, Ettore; Supuran, Claudiu T; Cosconati, Sandro; Taliani, Sabrina
A balance between elongation and trimming regulates telomere stability in stem cells 1-gen-2017 Rivera, Teresa; Haggblom, Candy; Cosconati, Sandro; Karlseder, Jan
A conformationally frozen peptoid boosts CXCR4 affinity and anti-HIV activity 1-gen-2012 Demmer, O; Frank, Ao; Hagn, F; Schottelius, M; Marinelli, L; Cosconati, Sandro; Brack Werner, R; Kremb, S; Wester, Hj; Kessler, H.
A more detailed picture of the interactions between virtual screening-derived hits and the DNA G-quadruplex: NMR, molecular modelling and ITC studies 1-gen-2011 Trotta, R; De Tito, S; Lauri, I; La Pietra, V; Marinelli, L; Cosconati, Sandro; Martino, L; Conte, Mr; Mayol, L; Novellino, E; Randazzo, A.
Antiproliferative and proapoptotic activity of CLM3, a novel multiple tyrosine kinase inhibitor, alone and in combination with SN-38 on endothelial and cancer cells 1-gen-2011 Bocci, G; Fioravanti, A; La Motta, C; Orlandi, P; Canu, B; Di Desidero, T; Mugnaini, L; Sartini, S; Cosconati, Sandro; Frati, R; Antonelli, A; Berti, P; Miccoli, P; Da Settimo, F; Danesi, R.
Antitumor efficacy of Kisspeptin in human malignant mesothelioma cells 1-gen-2018 Ciaramella, V; DELLA CORTE, CARMINIA MARIA; Di Mauro, C; Tomassi, S; Di Maro, S; Troiani, T; Martinelli, E; Bianco, R; Cosconati, S; Pierantoni, R; Meccariello, R; Chianese, R; Ciardiello, F; Morgillo, F.
Architecture of the human urotensin II receptor: Comparison of the binding domains of peptide and non-peptide urotensin II agonists 1-gen-2005 Lavecchia, A; Cosconati, Sandro; Novellino, E.
Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase 1-gen-2014 Costi, R; Metifiot, M; Chung, S; Crucitti, Gv; Maddali, K; Pescatori, L; Messore, A; Madia, Vn; Pupo, G; Scipione, L; Tortorella, S; Di Leva, Fs; Cosconati, Sandro; Marinelli, L; Novellino, E; Le Grice, Sfj; Corona, A; Pommier, Y; Marchand, C; Di Santo, R.
Benzofuroxane derivatives as multi-effective agents for the treatment of cardiovascular diabetic complications. Synthesis, functional evaluation, and molecular modeling studies 1-gen-2012 Sartini, S; Cosconati, Sandro; Marinelli, M; Barresi, E; DI MARO, Salvatore; Simorini, F; Taliani, S; Salerno, S; Marini, Am; Da Settimo, F; Novellino, E; La Motta, C.
Best Matching Protein Conformations and Docking Programs for a Virtual Screening Campaign Against SMO Receptor 1-gen-2016 Amendola, Giorgio; Dimaio, Danilo; Lapietra, Valeria; Cosconati, Sandro
Boosting Fmoc Solid-Phase Peptide Synthesis by Ultrasonication 1-gen-2019 Merlino, F.; Tomassi, S.; Yousif, A. M.; Messere, A.; Marinelli, L.; Grieco, P.; Novellino, E.; Cosconati, S.; Di Maro, S.
Carbonic anhydrase activation profile of indole-based derivatives 1-gen-2021 Barresi, E.; Ravichandran, R.; Germelli, L.; Angeli, A.; Baglini, E.; Salerno, S.; Marini, A. M.; Costa, B.; Da Pozzo, E.; Martini, C.; Da Settimo, F.; Supuran, C.; Cosconati, S.; Taliani, S.
Cationic nucleopeptides as novel non-covalent carriers for the delivery of peptide nucleic acid (PNA) and RNA oligomers 1-gen-2018 Tomassi, Stefano; Ieranò, Caterina; Mercurio, Maria Emilia; Nigro, Ersilia; Daniele, Aurora; Russo, Rosita; Chambery, Angela; Baglivo, Ilaria; Pedone, Paolo Vincenzo; Rea, Giuseppina; Napolitano, Maria; Scala, Stefania; Cosconati, Sandro; Marinelli, Luciana; Novellino, Ettore; Messere, Anna; Di Maro, Salvatore
Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic Activity 1-gen-2015 Eadsforth, Tc; Pinto, A; Luciani, R; Tamborini, L; Cullia, G; De Micheli, C; Marinelli, L; Cosconati, Sandro; Novellino, E; Lo Presti, L; Cordeiro da Silva, A; Conti, P; Hunter, Wn; Costi, M. P.
Characterizing the 1,4-dihydropyridines binding interactions in the L-type Ca2+ channel: Model construction and docking calculations 1-gen-2007 Cosconati, Sandro; Marinelli, L; Lavecchia, A; Novellino, E.
CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists 1-gen-2022 Tomassi, Stefano; Dimmito, Marilisa Pia; Cai, Minying; D'Aniello, Antonia; Del Bene, Alessandra; Messere, Anna; Liu, Zekun; Zhu, Tingyi; Hruby, Victor J; Stefanucci, Azzurra; Cosconati, Sandro; Mollica, Adriano; Di Maro, Salvatore
Computer-Aided Identification and Lead Optimization of Dual Murine Double Minute 2 and 4 Binders: Structure-Activity Relationship Studies and Pharmacological Activity 1-gen-2017 Giustiniano, Mariateresa; Daniele, Simona; Pelliccia, Sveva; La Pietra, Valeria; Pietrobono, Deborah; Brancaccio, Diego; Cosconati, Sandro; Messere, Anna; Giuntini, Stefano; Cerofolini, Linda; Fragai, Marco; Luchinat, Claudio; Taliani, Sabrina; La Regina, Giuseppe; Da Settimo, Federico; Silvestri, Romano; Martini, Claudia; Novellino, Ettore; Marinelli, Luciana