Sfoglia per Autore
1-methoxy-canthin-6-one and related β-carbolines: From natural compound to synthesis and biological activities
2012 Peduto, Antonella; Filosa, Rosanna; De Caprariis, Paolo; De Feo, Vincenzo; Li, Shiyou; Wang, Ping; De Martino, Laura
Active methylene compounds in a very effective approach to 3-substituted isobenzofuranones through tandem aldol/lactonization reactions
2012 Di Mola, Antonia; Croce, Gianluca; More, Vijaykumar; De Caprariis, Paolo; Filosa, Rosanna; Massa, Antonio
Synthesis and Reactivity of the 3-Substituted Isoindolinone Framework to Assemble Highly Functionalized Related Structures
2012 Petronzi, C; Collarile, S; Croce, G; Filosa, Rosanna; De Caprariis, P; Peduto, A; Palombi, L; Intintoli, V; Di Mola, A; Massa, A.
Cyclohexa-2,5-diene-1,4-dione-based antiproliferative agents: design, synthesis, and cytotoxic evaluation
2013 Petronzi, C; Festa, M; Peduto, A; Castellano, M; Marinello, J; Massa, A; Capasso, A; Capranico, G; LA GATTA, Annalisa; DE ROSA, Mario; Caraglia, Michele; Filosa, Rosanna
Design of inhibitors of influenza virus membrane fusion: Synthesis, structure-activity relationship and in vitro antiviral activity of a novel indole series.
2013 Brancato, V; Peduto, A; Wharton, S; Martin, S; More, V; Di Mola, A; Massa, A; Perfetto, Brunella; Donnarumma, Giovanna; Schiraldi, Chiara; Tufano, Ma; DE ROSA, Mario; Filosa, Rosanna; Hay, A.
Discovery and biological evaluation of novel 1,4-benzoquinone and related resorcinol derivatives that inhibit 5-lipoxygenase
2013 Filosa, Rosanna; Peduto, A; Aparoy, P; Schaible, Am; Luderer, S; Krauth, V; Petronzi, C; Massa, A; DE ROSA, Mario; Reddanna, P; Werz, O.
Potent inhibition of human 5-lipoxygenase and microsomal prostaglandin E-2 synthase-1 by the anti-carcinogenic and anti-inflammatory agent embelin
2013 Schaible, Am; Traber, H; Temml, V; Noha, Sm; Filosa, Rosanna; Peduto, A; Weinigel, C; Barz, D; Schuster, D; Werz, O.
Elucidation of the molecular mechanism and the efficacy in vivo of a novel 1,4-benzoquinone that inhibits 5-lipoxygenase.
2014 Schaible, Am; Filosa, Rosanna; Temml, V; Krauth, V; Matteis, M; Peduto, A; Bruno, F; Luderer, S; Roviezzo, F; Di Mola, A; de Rosa, M; D'Agostino, Bruno; Weinigel, C; Barz, D; Koeberle, A; Pergola, C; Schuster, D; Werz, O.
New chelating agents for Cu(II), Fe(III), Al(III), and Zn(II) based on beta-diketonate-3-substituted phthalide (isobenzofuranone) and isoindolinone
2014 Di Matteo, L; Christodoulakis, O; Filosa, Rosanna; De Caprariis, P; Di Mola, A; Vasca, E; Massa, A.
In vitro antiviral and immunomodulatory activity of arbidol and structurally related derivatives in herpes simplex virus type 1-infected human keratinocytes (HaCat).
2014 Perfetto, Brunella; Filosa, Rosanna; De Gregorio, V; Peduto, A; LA GATTA, Annalisa; de Caprariis, P; Tufano, Ma; Donnarumma, Giovanna
Further studies on ethyl 5-hydroxy-indole-3-carboxylate scaffold: Design, synthesis and evaluation of 2-phenylthiomethyl-indole derivatives as efficient inhibitors of human 5-lipoxygenase
2014 Peduto, A; Bruno, F; Dehm, F; Krauth, V; de Caprariis, P; Weinigel, C; Barz, D; Massa, A; DE ROSA, Mario; Werz, O; Filosa, Rosanna
Cascade reactions of glycine Schiff bases and chiral phase transfer catalysts in the synthesis of alpha-amino acids 3-substituted phthalides or isoindolinones
2014 Perillo, M; Di Mola, A; Filosa, Rosanna; Palombi, L; Massa, A.
Structure-activity relationship study of arbidol derivatives as inhibitors of chikungunya virus replication
2014 Di Mola, A; Peduto, A; LA GATTA, Annalisa; Delang, L; Pastorino, B; Neyts, J; Leyssen, P; DE ROSA, Mario; Filosa, Rosanna
Bifunctional phase-transfer catalysis in the asymmetric synthesis of biologically active isoindolinones
2015 Antonia Di Mola1, 2; Tiffner, Maximilian; Scorzelli, Francesco; Palombi, Laura; Filosa, Rosanna; Caprariis, Paolo De; Waser, Mario; Antonio, Massa
The Introduction of Inversion of Polarity Sites in DNA G-Quadruplex Structures: Effects and Perspectives
2015 Virgilio, A; Esposito, V; Filosa, Rosanna; Mayo, L; Galeone, A. 1.
3-Carboxylate Substituted Isoindolinones in K2CO3-Catalyzed Michael Reactions
2015 Scorzelli, F; Di Mola, A; Palombi, L; Filosa, Rosanna; Massa, A.
Novel series of benzoquinones with high potency against 5-lipoxygenase in human polymorphonuclear leukocytes
2015 Filosa, Rosanna; Peduto, A; Schaible, Am; Krauth, V; Weinigel, C; Barz, D; Petronzi, C; Bruno, F; Roviezzo, F; Spaziano, Giuseppe; D'Agostino, Bruno; DE ROSA, Mario; Werz, O.
Synthesis and pharmacological evaluation of functionalized isoindolinones on GABA-activated chloride currents in rat cerebellum granule cells in culture
2016 Di Mola, Antonia; Gatta, Elena; Petronzi, Carmen; Cupello, Aroldo; De Caprariis, Paolo; Robello, Mauro; Massa, Antonio; Filosa, Rosanna
Discovery of Novel multi-target Indole-based Derivatives as Potent and Selective Inhibitors of Chikungunya Virus Replication
2016 Scuotto, Maria; Abdelnabi, Rana; Collarile, Selene; Schiraldi, Chiara; Delang, Leen; Massa, Antonio; Ferla, Salvatore; Brancale, Andrea; Leyssen, Pieter; Neyts, Johan; Filosa, Rosanna
Optimization of hyaluronan-based eye drop formulations
2016 Salzillo, Rosanna; Schiraldi, Chiara; Corsuto, Luisana; D'Agostino, Antonella; Filosa, Rosanna; DE ROSA, Mario; LA GATTA, Annalisa
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
1-methoxy-canthin-6-one and related β-carbolines: From natural compound to synthesis and biological activities | 1-gen-2012 | Peduto, Antonella; Filosa, Rosanna; De Caprariis, Paolo; De Feo, Vincenzo; Li, Shiyou; Wang, Ping; De Martino, Laura | |
Active methylene compounds in a very effective approach to 3-substituted isobenzofuranones through tandem aldol/lactonization reactions | 1-gen-2012 | Di Mola, Antonia; Croce, Gianluca; More, Vijaykumar; De Caprariis, Paolo; Filosa, Rosanna; Massa, Antonio | |
Synthesis and Reactivity of the 3-Substituted Isoindolinone Framework to Assemble Highly Functionalized Related Structures | 1-gen-2012 | Petronzi, C; Collarile, S; Croce, G; Filosa, Rosanna; De Caprariis, P; Peduto, A; Palombi, L; Intintoli, V; Di Mola, A; Massa, A. | |
Cyclohexa-2,5-diene-1,4-dione-based antiproliferative agents: design, synthesis, and cytotoxic evaluation | 1-gen-2013 | Petronzi, C; Festa, M; Peduto, A; Castellano, M; Marinello, J; Massa, A; Capasso, A; Capranico, G; LA GATTA, Annalisa; DE ROSA, Mario; Caraglia, Michele; Filosa, Rosanna | |
Design of inhibitors of influenza virus membrane fusion: Synthesis, structure-activity relationship and in vitro antiviral activity of a novel indole series. | 1-gen-2013 | Brancato, V; Peduto, A; Wharton, S; Martin, S; More, V; Di Mola, A; Massa, A; Perfetto, Brunella; Donnarumma, Giovanna; Schiraldi, Chiara; Tufano, Ma; DE ROSA, Mario; Filosa, Rosanna; Hay, A. | |
Discovery and biological evaluation of novel 1,4-benzoquinone and related resorcinol derivatives that inhibit 5-lipoxygenase | 1-gen-2013 | Filosa, Rosanna; Peduto, A; Aparoy, P; Schaible, Am; Luderer, S; Krauth, V; Petronzi, C; Massa, A; DE ROSA, Mario; Reddanna, P; Werz, O. | |
Potent inhibition of human 5-lipoxygenase and microsomal prostaglandin E-2 synthase-1 by the anti-carcinogenic and anti-inflammatory agent embelin | 1-gen-2013 | Schaible, Am; Traber, H; Temml, V; Noha, Sm; Filosa, Rosanna; Peduto, A; Weinigel, C; Barz, D; Schuster, D; Werz, O. | |
Elucidation of the molecular mechanism and the efficacy in vivo of a novel 1,4-benzoquinone that inhibits 5-lipoxygenase. | 1-gen-2014 | Schaible, Am; Filosa, Rosanna; Temml, V; Krauth, V; Matteis, M; Peduto, A; Bruno, F; Luderer, S; Roviezzo, F; Di Mola, A; de Rosa, M; D'Agostino, Bruno; Weinigel, C; Barz, D; Koeberle, A; Pergola, C; Schuster, D; Werz, O. | |
New chelating agents for Cu(II), Fe(III), Al(III), and Zn(II) based on beta-diketonate-3-substituted phthalide (isobenzofuranone) and isoindolinone | 1-gen-2014 | Di Matteo, L; Christodoulakis, O; Filosa, Rosanna; De Caprariis, P; Di Mola, A; Vasca, E; Massa, A. | |
In vitro antiviral and immunomodulatory activity of arbidol and structurally related derivatives in herpes simplex virus type 1-infected human keratinocytes (HaCat). | 1-gen-2014 | Perfetto, Brunella; Filosa, Rosanna; De Gregorio, V; Peduto, A; LA GATTA, Annalisa; de Caprariis, P; Tufano, Ma; Donnarumma, Giovanna | |
Further studies on ethyl 5-hydroxy-indole-3-carboxylate scaffold: Design, synthesis and evaluation of 2-phenylthiomethyl-indole derivatives as efficient inhibitors of human 5-lipoxygenase | 1-gen-2014 | Peduto, A; Bruno, F; Dehm, F; Krauth, V; de Caprariis, P; Weinigel, C; Barz, D; Massa, A; DE ROSA, Mario; Werz, O; Filosa, Rosanna | |
Cascade reactions of glycine Schiff bases and chiral phase transfer catalysts in the synthesis of alpha-amino acids 3-substituted phthalides or isoindolinones | 1-gen-2014 | Perillo, M; Di Mola, A; Filosa, Rosanna; Palombi, L; Massa, A. | |
Structure-activity relationship study of arbidol derivatives as inhibitors of chikungunya virus replication | 1-gen-2014 | Di Mola, A; Peduto, A; LA GATTA, Annalisa; Delang, L; Pastorino, B; Neyts, J; Leyssen, P; DE ROSA, Mario; Filosa, Rosanna | |
Bifunctional phase-transfer catalysis in the asymmetric synthesis of biologically active isoindolinones | 1-gen-2015 | Antonia Di Mola1, 2; Tiffner, Maximilian; Scorzelli, Francesco; Palombi, Laura; Filosa, Rosanna; Caprariis, Paolo De; Waser, Mario; Antonio, Massa | |
The Introduction of Inversion of Polarity Sites in DNA G-Quadruplex Structures: Effects and Perspectives | 1-gen-2015 | Virgilio, A; Esposito, V; Filosa, Rosanna; Mayo, L; Galeone, A. 1. | |
3-Carboxylate Substituted Isoindolinones in K2CO3-Catalyzed Michael Reactions | 1-gen-2015 | Scorzelli, F; Di Mola, A; Palombi, L; Filosa, Rosanna; Massa, A. | |
Novel series of benzoquinones with high potency against 5-lipoxygenase in human polymorphonuclear leukocytes | 1-gen-2015 | Filosa, Rosanna; Peduto, A; Schaible, Am; Krauth, V; Weinigel, C; Barz, D; Petronzi, C; Bruno, F; Roviezzo, F; Spaziano, Giuseppe; D'Agostino, Bruno; DE ROSA, Mario; Werz, O.; Filosa, Rosanna; Peduto, A; Schaible, Am; Krauth, V; Weinigel, C; Barz, D; Petronzi, C; Bruno, F; Roviezzo, F; Spaziano, Giuseppe; D'Agostino, Bruno; DE ROSA, Mario; Werz, O. | |
Synthesis and pharmacological evaluation of functionalized isoindolinones on GABA-activated chloride currents in rat cerebellum granule cells in culture | 1-gen-2016 | Di Mola, Antonia; Gatta, Elena; Petronzi, Carmen; Cupello, Aroldo; De Caprariis, Paolo; Robello, Mauro; Massa, Antonio; Filosa, Rosanna | |
Discovery of Novel multi-target Indole-based Derivatives as Potent and Selective Inhibitors of Chikungunya Virus Replication | 1-gen-2016 | Scuotto, Maria; Abdelnabi, Rana; Collarile, Selene; Schiraldi, Chiara; Delang, Leen; Massa, Antonio; Ferla, Salvatore; Brancale, Andrea; Leyssen, Pieter; Neyts, Johan; Filosa, Rosanna | |
Optimization of hyaluronan-based eye drop formulations | 1-gen-2016 | Salzillo, Rosanna; Schiraldi, Chiara; Corsuto, Luisana; D'Agostino, Antonella; Filosa, Rosanna; DE ROSA, Mario; LA GATTA, Annalisa |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile