Sfoglia per Autore
Evaluation of alternative strategies to optimize ketorolac transdermal delivery
2006 Puglia, C; Filosa, Rosanna; Peduto, A; de Caprariis, P; Rizza, L; Bonina, F; Blasi, P.
Diastereoselectivity in the alkylation of 4-fluoroproline methyl esters
2006 Filosa, Rosanna; Holder, C; Auberson, Yp
Synthesis and biological evaluation of (2S)-and (2R)-2-(3 '-phosphonobicyclo[1.1.1]pentyl)glycines as novel group III selective metabotropic glutamate receptor ligands
2006 Filosa, Rosanna; Marinozzi, M; Costantino, G; Hermit, Mb; Thomsen, C; Pellicciari, R.
Synthesis and preliminary biological evaluation of 2 '-substituted 2-(3 '-carboxybicyclo[1.1.1]-pentyl)glycine derivatives as group I selective metabotropic glutamate receptor ligands
2006 :pellicciari, R; Filosa, Rosanna; Fulco, Mc; Marinozzi, M; Macchiarulo, A; Novak, C; Natalini, B; Hermit, Mb; Nielsen, S; Sager, Tn; Stensbol, Tb; Thomsen, C.
Synthesis and antiproliferative properties of N-3/8-disubstituted 3,8-diazabicyclo[3.2.1]octane analogues of 3,8-bis[2-(3,4,5-trimethoxyphenyl)pyridin-4-yl]methyl-piperazine
2007 Filosa, Rosanna; Peduto, A; de Caprariis, P; Saturnino, C; Festa, Maria; Petrella, A; Pau, A; Pinna, Ga; La Colla, P; Busonera, B; Loddo, R.
Molecular mechanism involved in the transport of a prodrug dopamine glycosyl conjugate
2007 Dalpiaz, A.; Filosa, Rosanna; de Caprariis, P.; Conte, G.; Bortolotti, F.; Biondi, C.; Scatturin, A.; Prasad, P. D.; Pavan, B.
Synthesis, physicochemical properties and in vitro permeation studies of new ketorolac ester derivatives.
2007 Puglia, Carmelo; Filosa, Rosanna; Peduto, Antonella; de Caprariis, Paolo; Boatto, Gianpiero; Nieddu, Maria; Santagati, Natale Alfredo; Bonina, Francesco
Antioxidant activity of diphenylpropionamide derivatives: Synthesis, biological evaluation and computational analysis
2008 Urbani, P; Ramunno, A; Filosa, Rosanna; Pinto, A; Popolo, A; Bianchino, E; Piotto, S; Saturnino, C; De Prisco, R; Nicolaus, B; Tommonaro, G.
A New Approach to Di- and Tetrasubstituted 2,3-Dihydropyridin-4(1H)-ones through Aza-Diels-Alder Reaction Promoted by Silicon Tetrachloride
2009 Massa, A; de Sio, V; Villano, R; Acocella, Mr; Palombi, L; Sellitto, G; Peduto, A; Filosa, Rosanna; De Capraris, P; Scettri, A.
Design, synthesis and biological evaluation of novel bicyclo[1.1.1] pentane-based omega-acidic amino acids as glutamate receptors ligands
2009 Filosa, Rosanna; Fulco, Mc; Marinozzi, M; Giacche, N; Macchiarulo, A; Peduto, A; Massa, A; de Caprariis, P; Thomsen, C; Christoffersen, C; Pellicciari, R.
Molecular modelling studies, synthesis and biological activity of a series of novel bisnaphthalimides and their development as new DNA topoisomerase II inhibitors
2009 Filosa, Rosanna; Peduto, A; Di Micco, S; de Caprariis, P; Festa, M; Petrella, A; Capranico, G; Bifulco, G.
Synthesis of beta-hydroxymalonates: the direct aldol addition of malonates to aldehydes in the presence of SiCl4 and i-Pr2EtN
2009 Massa, A; Scettri, A; Filosa, Rosanna; Capozzolo, L.
Trimethylchlorosilane and Silicon Tetrachloride in Two Novel Methodologies for the Efficient and Mild Aldol Addition of beta-Keto Esters and Malonates to Aldehydes
2010 Massa, A; Roscigno, A; De Caprariis, P; Filosa, Rosanna; Di Mola, A.
Synthesis and cytotoxic activity of new β-carboline derivatives
2011 Peduto, A; More, V; de Caprariis, P; Festa, M; Capasso, A; Piacente, S; De Martino, L; De Feo, V; Filosa, Rosanna
2,3-Dihydro-1,2-Diphenyl-substituted 4H-Pyridinone Derivatives as New Anti Flaviviridae Inhibitors
2011 Peduto, A; Massa, A; Di Mola, A; de Caprariis, P; La Colla, P; Loddo, R; Altamura, S; Maga, G; Filosa, Rosanna
Natural compounds in anti-leukaemic therapy: a review
2011 De Martino, L; D'Arena, G; Filosa, Rosanna; Peduto, A; Zeppa, R; De Feo, V.
Multi-component, regio-selective aldol addition of beta-ketoesters to aldehydes: scope and applications
2011 More, Vijaykumar; Di Mola, A; Croce, G; Tedesco, C; Petronzi, C; Peduto, A; De Caprariis, P; Filosa, Rosanna; Massa, A.
The aldol addition of readily enolizable 1,3-dicarbonyl compounds to 2-cyanobenzaldehyde in the synthesis of novel 3-substituted isoindolinones
2011 More, Vijaykumar; Dimola, Antonia; Perillo, Milena; Decaprariis, Paolo; Filosa, Rosanna; Peduto, Antonella; Massa, Antonio
Structure-based design, synthesis and preliminary anti-inflammatory activity of bolinaquinone analogues
2011 Petronzi, C; Filosa, Rosanna; Peduto, A; Monti, M; Margarucci, L; Massa, A; Ercolino, Sf; Bizzarro, V; Parente, L; Riccio, R; de Caprariis, P.
Design, synthesis, biophysical and biological studies of trisubstituted naphthalimides as G-quadruplex ligands
2011 Peduto, Antonella; Pagano, Bruno; Petronzi, Carmen; Massa, Antonio; Esposito, Veronica; Virgilio, Antonella; Paduano, Francesco; Trapasso, Francesco; Fiorito, Filomena; Florio, Salvatore; Giancola, Concetta; Galeone, Aldo; Filosa, Rosanna
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Evaluation of alternative strategies to optimize ketorolac transdermal delivery | 1-gen-2006 | Puglia, C; Filosa, Rosanna; Peduto, A; de Caprariis, P; Rizza, L; Bonina, F; Blasi, P. | |
Diastereoselectivity in the alkylation of 4-fluoroproline methyl esters | 1-gen-2006 | Filosa, Rosanna; Holder, C; Auberson, Yp | |
Synthesis and biological evaluation of (2S)-and (2R)-2-(3 '-phosphonobicyclo[1.1.1]pentyl)glycines as novel group III selective metabotropic glutamate receptor ligands | 1-gen-2006 | Filosa, Rosanna; Marinozzi, M; Costantino, G; Hermit, Mb; Thomsen, C; Pellicciari, R. | |
Synthesis and preliminary biological evaluation of 2 '-substituted 2-(3 '-carboxybicyclo[1.1.1]-pentyl)glycine derivatives as group I selective metabotropic glutamate receptor ligands | 1-gen-2006 | :pellicciari, R; Filosa, Rosanna; Fulco, Mc; Marinozzi, M; Macchiarulo, A; Novak, C; Natalini, B; Hermit, Mb; Nielsen, S; Sager, Tn; Stensbol, Tb; Thomsen, C. | |
Synthesis and antiproliferative properties of N-3/8-disubstituted 3,8-diazabicyclo[3.2.1]octane analogues of 3,8-bis[2-(3,4,5-trimethoxyphenyl)pyridin-4-yl]methyl-piperazine | 1-gen-2007 | Filosa, Rosanna; Peduto, A; de Caprariis, P; Saturnino, C; Festa, Maria; Petrella, A; Pau, A; Pinna, Ga; La Colla, P; Busonera, B; Loddo, R. | |
Molecular mechanism involved in the transport of a prodrug dopamine glycosyl conjugate | 1-gen-2007 | Dalpiaz, A.; Filosa, Rosanna; de Caprariis, P.; Conte, G.; Bortolotti, F.; Biondi, C.; Scatturin, A.; Prasad, P. D.; Pavan, B. | |
Synthesis, physicochemical properties and in vitro permeation studies of new ketorolac ester derivatives. | 1-gen-2007 | Puglia, Carmelo; Filosa, Rosanna; Peduto, Antonella; de Caprariis, Paolo; Boatto, Gianpiero; Nieddu, Maria; Santagati, Natale Alfredo; Bonina, Francesco | |
Antioxidant activity of diphenylpropionamide derivatives: Synthesis, biological evaluation and computational analysis | 1-gen-2008 | Urbani, P; Ramunno, A; Filosa, Rosanna; Pinto, A; Popolo, A; Bianchino, E; Piotto, S; Saturnino, C; De Prisco, R; Nicolaus, B; Tommonaro, G. | |
A New Approach to Di- and Tetrasubstituted 2,3-Dihydropyridin-4(1H)-ones through Aza-Diels-Alder Reaction Promoted by Silicon Tetrachloride | 1-gen-2009 | Massa, A; de Sio, V; Villano, R; Acocella, Mr; Palombi, L; Sellitto, G; Peduto, A; Filosa, Rosanna; De Capraris, P; Scettri, A. | |
Design, synthesis and biological evaluation of novel bicyclo[1.1.1] pentane-based omega-acidic amino acids as glutamate receptors ligands | 1-gen-2009 | Filosa, Rosanna; Fulco, Mc; Marinozzi, M; Giacche, N; Macchiarulo, A; Peduto, A; Massa, A; de Caprariis, P; Thomsen, C; Christoffersen, C; Pellicciari, R. | |
Molecular modelling studies, synthesis and biological activity of a series of novel bisnaphthalimides and their development as new DNA topoisomerase II inhibitors | 1-gen-2009 | Filosa, Rosanna; Peduto, A; Di Micco, S; de Caprariis, P; Festa, M; Petrella, A; Capranico, G; Bifulco, G. | |
Synthesis of beta-hydroxymalonates: the direct aldol addition of malonates to aldehydes in the presence of SiCl4 and i-Pr2EtN | 1-gen-2009 | Massa, A; Scettri, A; Filosa, Rosanna; Capozzolo, L. | |
Trimethylchlorosilane and Silicon Tetrachloride in Two Novel Methodologies for the Efficient and Mild Aldol Addition of beta-Keto Esters and Malonates to Aldehydes | 1-gen-2010 | Massa, A; Roscigno, A; De Caprariis, P; Filosa, Rosanna; Di Mola, A. | |
Synthesis and cytotoxic activity of new β-carboline derivatives | 1-gen-2011 | Peduto, A; More, V; de Caprariis, P; Festa, M; Capasso, A; Piacente, S; De Martino, L; De Feo, V; Filosa, Rosanna | |
2,3-Dihydro-1,2-Diphenyl-substituted 4H-Pyridinone Derivatives as New Anti Flaviviridae Inhibitors | 1-gen-2011 | Peduto, A; Massa, A; Di Mola, A; de Caprariis, P; La Colla, P; Loddo, R; Altamura, S; Maga, G; Filosa, Rosanna | |
Natural compounds in anti-leukaemic therapy: a review | 1-gen-2011 | De Martino, L; D'Arena, G; Filosa, Rosanna; Peduto, A; Zeppa, R; De Feo, V. | |
Multi-component, regio-selective aldol addition of beta-ketoesters to aldehydes: scope and applications | 1-gen-2011 | More, Vijaykumar; Di Mola, A; Croce, G; Tedesco, C; Petronzi, C; Peduto, A; De Caprariis, P; Filosa, Rosanna; Massa, A. | |
The aldol addition of readily enolizable 1,3-dicarbonyl compounds to 2-cyanobenzaldehyde in the synthesis of novel 3-substituted isoindolinones | 1-gen-2011 | More, Vijaykumar; Dimola, Antonia; Perillo, Milena; Decaprariis, Paolo; Filosa, Rosanna; Peduto, Antonella; Massa, Antonio | |
Structure-based design, synthesis and preliminary anti-inflammatory activity of bolinaquinone analogues | 1-gen-2011 | Petronzi, C; Filosa, Rosanna; Peduto, A; Monti, M; Margarucci, L; Massa, A; Ercolino, Sf; Bizzarro, V; Parente, L; Riccio, R; de Caprariis, P. | |
Design, synthesis, biophysical and biological studies of trisubstituted naphthalimides as G-quadruplex ligands | 1-gen-2011 | Peduto, Antonella; Pagano, Bruno; Petronzi, Carmen; Massa, Antonio; Esposito, Veronica; Virgilio, Antonella; Paduano, Francesco; Trapasso, Francesco; Fiorito, Filomena; Florio, Salvatore; Giancola, Concetta; Galeone, Aldo; Filosa, Rosanna |
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